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Study identifier: NCT03917043 Synced from ClinicalTrials.gov · July 29, 2026
● Recruiting

APG-2449 in Patients With Advanced Solid Tumors

Condition: Advanced Solid Cancer · Non Small Cell Lung Cancer · Esophageal Cancer  ·  Sponsor: Ascentage Pharma Group Inc.

PhasePhase 1
Planned participants165
Who can joinAll sexes, 18 Years to no upper limit
Healthy volunteersNo

About this study

APG-2449 is a novel, orally active, multi-targeted tyrosine kinase inhibitor, which inhibits FAK, ALK, and ROS1 with nanomolar potencies. In preclinical studies, APG-2449 demonstrated potent antiproliferative activity in various cancer cell lines as a single agent. In combination treatment, APG-2449 enhanced anti-proliferative activities of several chemotherapeutic and targeted agents. It is indicated that APG-2449 may have a broad therapeutic potential for the treatment of human cancer as a single agent and in combination with other classes of anticancer drugs. APG-2449 is intended for the treatment of patients with advanced solid tumors. Upon completion of the Phase 1 dose escalation study to establish the maximum tolerated dose (MTD), dose-limiting toxicities (DLTs), and/or recommended phase 2 dose (RP2D), several phase Ib/II studies will be implemented accordingly.

This description comes directly from the study's public registry record.

Talk to the study team

Yifan Zhai, M.D., Ph.D.  ·  +86-20-28069260  ·  yzhai@ascentage.com

Always discuss trial participation with your own doctor first.

Locations (9)

Beijing Cancer HospitalBeijing, Beijing Municipality, ChinaRecruiting
Fujian Medical University Union HospitalFuzhou, Fujian, ChinaNot Yet Recruiting
Fujian Cancer HospitalFuzhou, Fujian, ChinaNot Yet Recruiting
Sun-Yat Sen University Cancer CenterGuangzhou, Guangdong, ChinaRecruiting
The First affiliated hospital, Sun Yat-sen UniversityGuangzhou, Guangdong, ChinaRecruiting
Henan Provincial Oncology HospitalZhengzhou, Henan, ChinaRecruiting
Union Hospital medical college Huazhong University of Science and TechnologyWuhan, Hubei, ChinaRecruiting
Hunan Provincial Oncology HospitalChangsha, Hunan, ChinaRecruiting
Zhejiang Provincial Oncology HospitalHangzhou, Zhejiang, ChinaRecruiting

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Source record: clinicaltrials.gov/study/NCT03917043